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Safety and pharmacokinetics evaluation study according to the dose of camostat mesylate in healthy volunteers
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| Label | Type | Description | Intervention Names |
|---|---|---|---|
| Cohort 1 (Part 1) | Experimental | DWJ1248 100mg (100mg 1tab) PO |
|
| Cohort 2 (Part 1) | Experimental | DWJ1248 200mg (100mg 2tab) PO |
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| Cohort 3 (Part 1) | Experimental | DWJ1248 300mg (100mg 3tab) PO |
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| Group A (Part 2) | Experimental | DWJ1248 100mg 2tab PO - Wash out - DWJ1248 200mg 1tab PO |
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| Group B (Part 2) | Experimental | DWJ1248 200mg 1tab PO - Wash out - DWJ1248 100mg 2tab PO |
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| Name | Type | Description | Arm Group Labels | Other Names |
|---|---|---|---|---|
| DWJ1248 | Drug | Camostat mesylate Tablet from Daewoong |
|
| Measure | Description | Time Frame |
|---|---|---|
| Cmax of GBPA | Maximum blood concentration of GBPA (GUANIDINO BENZOYLOXY PHENYLACETIC ACID METHANESULFONATE) among observed blood concentrations at time points
| 0-6 hr |
| AUClast of GBPA | Area under the blood concentration-time of GBPA (GUANIDINO BENZOYLOXY PHENYLACETIC ACID METHANESULFONATE) among observed blood concentrations at time points
| 0-6 hr |
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Inclusion Criteria:
Exclusion Criteria:
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| Facility | Status | City | State | ZIP | Country | Contacts |
|---|---|---|---|---|---|---|
| Chungnam National University Hospital | Daejeon | 35015 | South Korea |
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Part1. Parallel, Part2. Crossover
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